Incorporation of water-solubilizing groups in pyrazolopyrimidine mTOR inhibitors: Discovery of highly potent and selective analogs with improved human microsomal stability
Author:
David J. Richard,Jeroen C. Verheijen,Kevin Curran,Joshua Kaplan,Lourdes Toral-Barza,Irwin Hollander,Judy Lucas,Ker Yu,Arie Zask
Publication:
Bioorganic & Medicinal Chemistry Letters
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